A new synthesis and preliminary evaluation of some analogues of mecamylamine - a compound with anti-addiction properties.
نویسندگان
چکیده
A new synthesis of mecamylamine - a known anti-hypertensive drug with anti-addictive properties is described. The new route allowed access to two novel analogues whose activity at two nicotinic acetylcholine receptor subtypes was assessed.
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 14 46 شماره
صفحات -
تاریخ انتشار 2016